Asymmetric Synthesis of Nitrogen Heterocycles (eBook)

Jacques Royer is Director of Research at the CNRS. He is currently the head of a laboratory of medicinal chemistry at the University Paris Descartes. He got his PhD at the University of Paris-Sud Orsay, and worked for 18 years at the Institut de Chimie des Substances Naturelles at the CNRS in Gif-sur-Yvette in the group of Prof. Henri-Philippe Husson. His research areas are asymmetric synthesis of natural products and more particularly alkaloids, amino alcohols and amino acids as well as original methods of synthesis including electrosynthesis. He is the author of about 100 publications in international renowned journals.

PART 1: Asymmetric Synthesis of Nitrogen Heterocycles Containing Only One Heteroatom

ASYMMETRIC SYNTHESIS OF THREE- AND FOUR-MEMBERED RING HETEROCYCLES
Substituted Aziridines
Substituted Monocyclic Azetidines and Carbocyclic-Fused Systems
ASYMMETRIC SYNTHESIS OF FIVE-MEMBERED RING HETEROCYCLES
Monocyclic Pyrrolidines and Pyrrolidinones
Pyrrolines
Fused Bicyclic Systems with Bridgehead Nitrogen
ASYMMETRIC SYNTHESIS OF SIX-MEMBERED RING HETEROCYCLES
Introduction
Dihydropyridines
Tetrahydropyridines
Monocyclic Piperidines and Carbocyclic Fused Systems
Fused Tri- or Bicyclic System with Bridgehead Nitrogen
ASYMMETRIC SYNTHESIS OF SEVEN- AND MORE-MEMBERED RING HETEROCYCLES
Substituted Azepines
Substituted Azocines
Substituted Large Nitrogen-Containing Rings

PART 2: Asymmetric Synthesis of Nitrogen Heterocycles With More Than One Heteroatom

ASYMMETRIC SYNTHESIS OF THREE- AND FOUR-MEMBERED RING HETEROCYCLES WITH MORE THAN ONE HETEROATOM
Introduction
Three-Membered N-Heterocycles with Two Heteroatoms
Four-Membered N-Heterocycles with Two Heteroatoms
ASYMMETRIC SYNTHESIS OF FIVE-MEMBERED RING HETEROCYCLES WITH MORE THAN ONE HETEROATOM
Five-Membered Heterocycles with N and O Atoms
Five-Membered Heterocycles with Two N Atoms
Five-Membered Heterocycles with N and S Atoms
ASYMMETRIC SYNTHESIS OF SIX-MEMBERED RING NITROGEN HETEROCYCLES WITH MORE THAN ONE HETEROATOM
Six-Membered Rings with Another Heteroatom in the Same Ring
ASYMMETRIC SYNTHESIS OF SEVEN-MEMBERED RINGS WITH MORE THAN ONE HETEROATOM
Diazepines
Oxazepines
Thiazepines